SURE

Article

Borrello, Maria Teresa, Benelkebir, Hanae, Lee, Adam, Tam, Chak Hin, Shafat, Manar, Rushworth, Stuart A, Bowles, Kristian A, Douglas, Leon, Duriez, Patrick J, Bailey, Sarah, Crabb, Simon J, Packham, Graham and Ganesan, A (2021) Synthesis of Carboxamide-Containing Tranylcypromine Analogues as LSD1 (KDM1A) Inhibitors Targeting Acute Myeloid Leukemia. ChemMedChem, 16. pp. 1316-1324. ISSN 1860-7187

Lecointre, Bertrand, Narozny, Remy, Borrello, Maria Teresa, Senger, Johanna, Alokta, Chakrabarti, Manfred, Jung, Marek, Martin, Romier, Christophe, Melesina, Jelena, Sippl, Wolfgang, Bischoff, Laurent and Ganesan, A (2018) Isoform-selective HDAC1/6/8 inhibitors with an imidazo-ketopiperazine cap containing stereochemical diversity. Philosophical transactions of the Royal Society B. ISSN 0962-8436

Borrello, Maria Teresa, Schinor, Benjamin, Bartels, Katharina, Benelkebir, Hanae, Pereira, Sara, Al-Jamal, Wafa T, Douglas, Leon, Duriez, Patrick J, Packham, Graham, Haufe, Gunter and Ganesan, A (2017) Fluorinated tranylcypromine analogues as inhibitors of lysine-specific deme-thylase 1 (LSD1, KDM1A. Bioorganic and Medicinal Chemistry Letters, 27 (10). pp. 2099-2101. ISSN 0960-894X

Book Section

Lee, Adam, Borrello, Maria Teresa and Ganesan, A (2019) LSD (Lysine-Specific Demethylase): A Decade-Long Trip from Discovery to Clinical Trials. In: Epigenetic Drug Discovery. Methods and Principles in Medicinal Chemistry, 1 . Wiley‐VCH Verlag GmbH & Co. KGaA, pp. 221-261. ISBN 9783527809257