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Abdelkader, Dalia H., El-Gizawy, Sanaa A., Faheem, Ahmed, McCarron, Paul A. and Osman, Mohamed A. (2018) Effect of process variables on formulation, in-vitro characterisation and subcutaneous delivery of insulin PLGA nanoparticles: An optimisation study. Journal of Drug Delivery Science and Technology, 43. pp. 160-171. ISSN 17732247

Abeke, Egega (2017) Dietary Analysis of Barley Crop for Animal Feed Supplementation in Poultry Farming. Doctoral thesis, University of Sunderland.

Andersen, O.A., Nathubhai, Amit, Dixon, M.J., Eggleston, I.M. and van Aalten, D.M.F. (2008) Structure-Based Dissection of the Natural Product Cyclopentapeptide Chitinase Inhibitor Argifin. Chemistry & Biology, 15 (3). pp. 295-301. ISSN 1074-5521

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Cherian, Thomas (2014) A Functional Study of the Ureter: Relevance of Myogenic and Neurogenic Functions and the Role of Post-Synaptic Alpha 1 and Alpha 2 Adrenergic Recepters in Ureteral Motility. Doctoral thesis, University of Sunderland.

Childs, Stephen, Haroune, Nicolas, Williams, Lee and Gronow, Michael (2017) Investigation of the Low Molecular Weight Thiol Composition in a Metastatic Prostate Cancer Cell Line (LNCaP) by LC-UV-MS and NMR after Labelling with the Ellman Reagent. American Journal of Analytical Chemistry, 08 (01). pp. 1-18. ISSN 2156-8251

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Dixon, M.J., Andersen, O.A., van Aalten, D. M. F., Nathubhai, Amit and Eggleston, I.M. (2007) Cyclic peptide chitinase inhibitors: New leads for antifungal and anti-inflammatory drugs. Biopolymers, 88 (4). p. 576. ISSN 0006-3525

Dixon, M.J., Andersen, O.A., van Aalten, D.M.F., Nathubhai, Amit and Eggleston, I.M. (2008) Synthesis of cyclic peptide chitinase inhibitors: Natural products with chemotherapeutic potential. Journal of Peptide Science, 14 (8). p. 13. ISSN 1075-2617

Dixon, M.J., Giuntini, F., Nathubhai, Amit, Andersen, O.A., van Aalten, D.M.F. and Eggleston, I.M. (2008) Synthetic approaches to cyclic peptide natural products as chitinase inhibitors. Journal of Peptide Science, 14 (8). p. 55. ISSN 1075-2617

Dixon, M.J., Nathubhai, Amit, Andersen, O.A., van Aalten, D.M.F. and Eggleston, I.M. (2008) Solid-phase synthesis of cyclic peptide chitinase inhibitors: SAR of the argifin scaffold. Organic & Biomolecular Chemistry, 7. pp. 259-268. ISSN 1477-0520

Dixon, M.J., Nathubhai, Amit, Andersen, O.A., van Aalten, D.M.F. and Eggleston, I.M. (2009) Synthesis and structure-based dissection of cyclic peptide chitinase inhibitors: New leads for antifungal and anti-inflammatory drugs. Advances in Experimental Medicine and Biology, 611. pp. 525-526. ISSN 0065-2598

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Elkordy, Amal, Forbes, Robert T and Barry, Brian W (2008) Study of protein conformational stability and integrity using calorimetry and FT-Raman spectroscopy correlated with enzymatic activity. European Journal of Pharmaceutical Sciences, 33 (2). pp. 177-190. ISSN 0928-0987

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Fatouros, Dimitrios, Douroumis, D, Nikolakis, V, Ntais, S, Moschovi, Anastasia Maria, Trivedi, V, Khima, B, Roldo, Marta, Nazar, Hamde and Cox, Paul (2011) In vitro and in silico investigations of drug delivery via zeolite BEA. Journal of Materials Chemistry (21). pp. 7789-7794. ISSN 0959-9428

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Khattab, RA, Elbandy, M, Lawrence, A, Paget, Timothy, Rae-Rho, J, Binnaser, YS and Ali, I (2018) Extraction, identification and biological activities of saponins in sea cucumber Pearsonothuria graeffei. Comb Chem High Throughput Screen, 21 (3). pp. 222-231. ISSN 1386-2073

Kumpan, K., Nathubhai, Amit, Zhang, C., Wood, P.J., Lloyd, M.D., Thompson, A.S., Haikarainen, T., Lehtiö, L. and Threadgill, M.D. (2015) Structure-based design, synthesis and evaluation in vitro of arylnaphthyridinones, arylpyridopyrimidinones and their tetrahydro derivatives as inhibitors of the tankyrases. Bioorganic & Medicinal Chemistry, 23. pp. 3013-3032. ISSN 0968-0896

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Mahita, Mwajuma, Abuhamdah, Rushdie, Howes, Melanie-Jayne, Ennaceur, Abdelkader, Abuhamdah, S and Chazot, Paul (2014) Identification of a Novel GABAA Receptor Channel Ligand Derived from Melissa officinalis and Lavandula angustifolia Essential Oils. European Journal of Medicinal Plants, 4 (7). pp. 810-818. ISSN 2231-0894

McGarry, Kenneth and Assamoha, Ennock (2017) Data integration with self-organising neural network reveals chemical structure and therapeutic effects of drug ATC codes. In: The 17th Annual UK Workshop on Computational Intelligence (UKCI-2017), 6-8 Sep 2017, Cardiff. (In Press)

McGarry, Kenneth, Graham, Yitka, McDonald, Sharon and Rashid, Anuam (2018) RESKO: Repositioning drugs by using side effects and knowledge from ontologies. Knowledge-Based Systems. pp. 34-48. ISSN 09507051

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Nathubhai, Amit, Haikarainen, T, Hayward, P.C., Munoz-Descalzo, S., Thompson, A.S., Lloyd, M.D., Lehtio, L. and Threadgill, M.D. (2016) Structure-activity relationships of 2-arylquinazolin-4-ones as highly selective and potent inhibitors of the tankyrases. European Journal of Medicinal Chemistry, 118. pp. 316-327. ISSN 0223-5234

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Nathubhai, Amit, Patterson, R., Woodman, T.J., Sharp, H.E.C., Chui, M.T.Y., Chung, H.H.K., Lau, W.S., Zheng, J., Lloyd, M.D., Thompson, A.S. and Threadgill, M.D. (2011) N3-Alkylation during formation of quinazolin-4-ones from condensation of anthranilamides and orthoamides. Organic & Biomolecular Chemistry, 9. pp. 6089-6099. ISSN 1477-0520

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Nathubhai, Amit, Wood, P.J., Lloyd, M.D., Thompson, A.S. and Threadgill, M.D. (2013) Design and Discovery of 2‑Arylquinazolin-4-ones as Potent and Selective Inhibitors of Tankyrases. ACS Medicinal Chemistry Letters, 4 (12). pp. 1173-1177. ISSN 1948-5875

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Ousset, Aymeric, Chavez, Pierre-François, Meeus, Joke, Robin, Florent, Schubert, Martin Alexander, Somville, Pascal and Dodou, Kalliopi (2018) Prediction of Phase Behavior of Spray-Dried Amorphous Solid Dispersions: Assessment of Thermodynamic Models, Standard Screening Methods and a Novel Atomization Screening Device with Regard to Prediction Accuracy. Pharmaceutics, 10 (1). pp. 29-54. ISSN 1999-4923; CODEN: PHARK5

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Paget, Timothy (2017) The Chemical Characterization of Nigerian Propolis samples and Their Activity Against Trypanosoma brucei. Scientific reports, 7 (923). ISSN 2045-2322

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Varadi, Linda, Gray, Mark, Groundwater, Paul, Hall, Andrew, James, Arthur L, Orenga, Sylvain, Perry, John D and Anderson, Rosaleen (2012) Synthesis and evaluation of fluorogenic 2-amino-1,8-naphthyridine derivatives for the detection of bacteria. Organic & Biomolecular Chemistry, 10 (13). pp. 2578-2589. ISSN 1477-0520

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Yevglevskis, M., Lee, G. L, Nathubhai, Amit, Petrova, Y.D., James, T.D., Threadgill, M.D., Woodman, T.J and Lloyd, M.D. (2018) Structure-activity relationships of rationally designed AMACR 1A inhibitors. BIOORGANIC CHEMISTRY, 79. pp. 145-154. ISSN 0045-2068

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Zaytsev, Andrey V, Anderson, Rosaleen, Bedernjak, Alexandre, Groundwater, Paul, Huang, Yongxue and Perry, John D (2008) Synthesis and testing of chromogenic phenoxazinone substrates for β-alanyl aminopeptidase. Organic and Biomolecular Chemistry, 6 (4). pp. 682-692. ISSN 1477-0520

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